Compounds > trapoxin a
Page last updated: 2024-09-03

trapoxin a and (3S,6S,9S,12R)-3-[(2S)-Butan-2-yl]-6-[(1-methoxyindol-3-yl)methyl]-9-(6-oxooctyl)-1,4,7,10-tetrazabicyclo[10.4.0]hexadecane-2,5,8,11-tetrone

trapoxin a has been researched along with (3S,6S,9S,12R)-3-[(2S)-Butan-2-yl]-6-[(1-methoxyindol-3-yl)methyl]-9-(6-oxooctyl)-1,4,7,10-tetrazabicyclo[10.4.0]hexadecane-2,5,8,11-tetrone in 1 studies

Compound Research Comparison

Studies
(trapoxin a)		Trials
(trapoxin a)		Recent Studies (post-2010)
(trapoxin a)		Studies
((3S,6S,9S,12R)-3-[(2S)-Butan-2-yl]-6-[(1-methoxyindol-3-yl)methyl]-9-(6-oxooctyl)-1,4,7,10-tetrazabicyclo[10.4.0]hexadecane-2,5,8,11-tetrone)		Trials
((3S,6S,9S,12R)-3-[(2S)-Butan-2-yl]-6-[(1-methoxyindol-3-yl)methyl]-9-(6-oxooctyl)-1,4,7,10-tetrazabicyclo[10.4.0]hexadecane-2,5,8,11-tetrone)		Recent Studies (post-2010) ((3S,6S,9S,12R)-3-[(2S)-Butan-2-yl]-6-[(1-methoxyindol-3-yl)methyl]-9-(6-oxooctyl)-1,4,7,10-tetrazabicyclo[10.4.0]hexadecane-2,5,8,11-tetrone)
80138115

Protein Interaction Comparison

ProteinTaxonomytrapoxin a (IC50)(3S,6S,9S,12R)-3-[(2S)-Butan-2-yl]-6-[(1-methoxyindol-3-yl)methyl]-9-(6-oxooctyl)-1,4,7,10-tetrazabicyclo[10.4.0]hexadecane-2,5,8,11-tetrone (IC50)
Histone deacetylase 3Homo sapiens (human)0.0151
Cytochrome P450 1A2Homo sapiens (human)0.011
Cytochrome P450 3A4Homo sapiens (human)0.011
Cytochrome P450 2D6Homo sapiens (human)0.034
Cytochrome P450 2C9 Homo sapiens (human)0.034
Tissue factorHomo sapiens (human)0.175
Cytochrome P450 2B6Homo sapiens (human)0.034
Cytochrome P450 3A5Homo sapiens (human)0.011
Cytochrome P450 2C19Homo sapiens (human)0.011
Histone deacetylase 4Homo sapiens (human)1.0335
Histone deacetylase 1Homo sapiens (human)0.0227
Histone deacetylase 7Homo sapiens (human)0.014
Histone deacetylase 2Homo sapiens (human)0.0185
Polyamine deacetylase HDAC10Homo sapiens (human)0.014
Histone deacetylase 11 Homo sapiens (human)0.014
Histone deacetylase 8Homo sapiens (human)0.2852
Histone deacetylase Cryptosporidium parvum0.001
Histone deacetylase Cryptosporidium parvum0.001
Histone deacetylase 6Homo sapiens (human)1.4663
Histone deacetylase 9Homo sapiens (human)0.014
Histone deacetylase 5Homo sapiens (human)0.014
Histone deacetylase Plasmodium falciparum (malaria parasite P. falciparum)0.001
Nuclear receptor corepressor 2Homo sapiens (human)0.0193

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chou, CJ; Gottesfeld, JM; Hu, F1

Other Studies

1 other study(ies) available for trapoxin a and (3S,6S,9S,12R)-3-[(2S)-Butan-2-yl]-6-[(1-methoxyindol-3-yl)methyl]-9-(6-oxooctyl)-1,4,7,10-tetrazabicyclo[10.4.0]hexadecane-2,5,8,11-tetrone

ArticleYear
Design and synthesis of novel hybrid benzamide-peptide histone deacetylase inhibitors.
    Bioorganic & medicinal chemistry letters, 2009, Jul-15, Volume: 19, Issue:14

    Topics: Benzamides; Cyclization; Drug Design; Enzyme Inhibitors; Histone Deacetylase 1; Histone Deacetylase Inhibitors; Histone Deacetylases; Humans; Neuroprotective Agents; Peptides

2009